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★★★★★
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Hire Dr. Kalpana T.
India

PhD in Pharmaceutical Chemistry experienced in writing and publishing 21 scientific articles in reputed journals.

Profile Summary
Subject Matter Expertise
Services
Writing Technical Writing
Research Market Research, User Research, Meta-Research, Feasibility Study, Gap Analysis, Gray Literature Search, Systematic Literature Review, Secondary Data Collection
Data & AI Statistical Analysis
Work Experience

Assistant Professor

Bharati Vidyapeeth's College of Pharmacy

January 2021 - Present

PhD student & Research Fellow

Bharati Vidyapeeth's College of Pharmacy

September 2017 - January 2021

Education

PhD

Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, India

January 2017 - January 2021

Certifications
  • Certification details not provided.
Publications
JOURNAL ARTICLE
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes(2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals. 14. (10). p. 1032. {MDPI} {AG}
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes (2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals.
Upadhyay, N., Tilekar, K., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Meyer-Almes, F.-J., Pokrovsky, V.S., et al.(2021). Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy . Bioorganic Chemistry. 107.
Kalpana Tilekar, Neha Upadhyay, Jessica D. Hess, Lucasantiago Henze Macias, Piotr Mrowka, Renato J. Aguilera, Franz-Josef Meyer-Almes, Cristina V. Iancu, Jun-yong Choe, C.S. Ramaa(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202. p. 112603. Elsevier {BV}
Tilekar, K., Upadhyay, N., Meyer-Almes, F.-J., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Pokrovsky, V.S., et al.(2020). Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents . ChemMedChem. 15. (19). p. 1813-1825.
Tilekar, K., Upadhyay, N., Hess, J.D., Macias, L.H., Mrowka, P., Aguilera, R.J., Meyer-Almes, F.-J., Iancu, C.V., Choe, J.-Y., Ramaa, C.S.(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202.
Tilekar, K., Upadhyay, N., Jänsch, N., Schweipert, M., Mrowka, P., Meyer-Almes, F.J., Ramaa, C.S.(2020). Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines . Bioorganic Chemistry. 95.
Joshi, H., Patil, V., Tilekar, K., Upadhyay, N., Gota, V., Ramaa, C.S.(2020). Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib . Bioorganic and Medicinal Chemistry Letters. 30. (23).
Upadhyay, N., Tilekar, K., Jänsch, N., Schweipert, M., Hess, J.D., Henze Macias, L., Mrowka, P., Aguilera, R.J., Choe, J.-Y., Meyer-Almes, F.-J., et al.(2020). Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation . Bioorganic Chemistry. 100.
Tilekar, K., Upadhyay, N., Schweipert, M., Hess, J.D., Macias, L.H., Mrowka, P., Meyer-Almes, F.-J., Aguilera, R.J., Iancu, C.V., Choe, J.-Y., et al.(2020). Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells . European Journal of Pharmaceutical Sciences. 154.
Tilekar, K., Upadhyay, N., Iancu, C.V., Pokrovsky, V., Choe, J.-Y., Ramaa, C.S.(2020). Power of two: combination of therapeutic approaches involving glucose transporter (GLUT) inhibitors to combat cancer . Biochimica et Biophysica Acta - Reviews on Cancer. 1874. (2).
Vora, D., Upadhyay, N., Tilekar, K., Jain, V., Ramaa, C.S.(2019). Development of 1,2,4-triazole-5-thione derivatives as potential inhibitors of enoyl acyl carrier protein reductase (Inha) in tuberculosis . Iranian Journal of Pharmaceutical Research. 18. (4). p. 1742-1758.
Kabir, A., Tilekar, K., Upadhyay, N., Ramaa, C.S.(2018). Novel anthraquinone derivatives as dual inhibitors of topoisomeras e 2 and casein kinase 2: In silico studies, synthesis and biological evaluation on leukemic cell lines . Anti-Cancer Agents in Medicinal Chemistry. 18. (11). p. 1551-1562.
Patil, V., Tilekar, K., Mehendale-Munj, S., Mohan, R., Ramaa, C.S.(2010). Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2,4- thiazolidinedione derivatives . European Journal of Medicinal Chemistry. 45. (10). p. 4539-4544.
Ramaa, C.S., Tilekar, K.N., Patil, V.M.(2010). Liver cancer: Different approaches for targeting . International Journal of PharmTech Research. 2. (1). p. 834-842.